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Analysis of the influence of selected thiosemicarbazides, 1,2,4-triazoles and 1,3,4-thiadiazoles’ structure on their microbiological activity against Candida Albicans ATCC30028 and Candida Albicans clinical isolate 26

  • Medical University of Warsaw

Research output: Chapter in Book/Report/Conference proceedingConference contributionpeer-review

Abstract

Considering the increasing incidence of fungal infections, in silico research of selected thiosemicarbazides, 1,2,4-triazoles and 1,3,4-thiadiazoles exhibiting varied biological activity against the Candida albicans fungi has been conducted in relation to this paper. The determined molecular descriptors for all 30 examined compounds and the published microbiological research served as the basis for obtaining multilinear QSAR models describing the relationship between biological activity against the Candida albicans ATCC 30028 and Candida albicans clinical isolate 26 fungi and the structure of examined compounds. The Leave-One-Out Cross Validation method was used to verify obtained models. The obtained Quantitative Structure-Activity Relationships are characterized by high determination coefficients and good prediction power. Additionally, the results of cluster analysis of compounds on the basis of their physicochemical parameters have also been presented.

Original languageEnglish
Title of host publicationInnovations in Biomedical Engineering, IBE 2018
EditorsEwaryst Tkacz, Marek Gzik, Zbigniew Paszenda, Ewa Pietka
PublisherSpringer Verlag
Pages149-158
Number of pages10
ISBN (Print)9783030154714
DOIs
Publication statusPublished - 2019
EventConference on Innovations in Biomedical Engineering, IBE 2018 - Katowice, Poland
Duration: 18 Oct 201820 Oct 2018

Publication series

NameAdvances in Intelligent Systems and Computing
Volume925
ISSN (Print)2194-5357
ISSN (Electronic)2194-5365

Conference

ConferenceConference on Innovations in Biomedical Engineering, IBE 2018
Country/TerritoryPoland
CityKatowice
Period18/10/1820/10/18

Keywords

  • 1, 2, 4 -triazoles
  • 1, 3, 4 -thiadiazoles
  • Cluster analysis
  • Multiple linear regression
  • Quantitative Structure-Activity Relationship
  • Thiosemicarbazides

ASJC Scopus subject areas

  • Control and Systems Engineering
  • General Computer Science

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